APIM050248: TGX-221
CAS No.: 663619-89-4.
Purity: >99% (HPLC at 214 and 254 nm).
QC: LC/MS, 1HNMR.
Solubility: Soluble in DMSO and Alcohols.APIM050249: TORIN 2
CAS No.: 1223001-51-1.
Purity: 99.9% by HPLC at 214 and 254 nm.
QC: HPLC-MS, 1H-NMR, and Quantitative Elemental Analysis Report.
Solubility: Refer to Certificate of Analysis.APIM050250: ULIXERTINIB (BVD-523, VRT752271)
CAS No.: 869886-67-9.
Purity: 100% optical purity (Chiral HPLC), 99.5% chemical purity (HPLC at 214 and 254 nm).
QC: HPLC-MS, 1HNMR, Chiral HPLC and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.APIM050251: UPROSERTIB (GSK2141795)
CAS No.: 1047634-65-0 (free base) 1047635-80-2 (HCl salt).
Purity: 99.5% chem purity (HPLC at 214 and 254 nm), 100% optical purity (Chiral HPLC), [α]20D = +5.4 o (c 1.0, MeOH).
QC: HPLC-MS, 1HNMR, Chiral HPLC, and Quantitative Elemental Analysis Report.
Solubility: Soluble in DMSO.APIM050252: VANDETANIB
CAS No.: 443913-73-3.
Purity: >99% (HPLC).
QC: 1HNMR, HPLC.
Solubility: Soluble in DMSO.APIM050253: VATALANIB
CAS No.: 212141-54-3.
Purity: >99% (HPLC).
QC: 1HNMR, HPLC.
Solubility: Soluble in water.APIM050254: VE-822 (BERZOSERTIB)
CAS No.: 1232416-25-9.
Purity: >99.5% (HPLC at 214 and 254 nm).
QC: HPLC-MS, 1HNMR, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.APIM050255: VOLITINIB (AZD6094, SAVOLITINIB)
CAS No.: 1313725-88-0.
Purity: 100% optical purity (Chiral HPLC), 99.8% chemical purity (HPLC at 215 and 254 nm).
QC: HPLC-MS, 1HNMR, Chiral HPLC, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO (22.7mg/ml, 50mM).APIM050313: AZD3965
CAS No.: 1448671-31-5.
Purity: >99% (HPLC at 214 and 254 nm), >98.5% Optical Purity (Chiral HPLC).
QC: HPLC-MS, 1HNMR, Chiral HPLC, and Quantitative Elemental Analysis.
Solubility: Soluble in DMSO.APIM050257: VS-4718 (PND-1186)
CAS No.: 1061353-68-1.
Purity: 99.9% (HPLC at 214 and 254 nm).
QC: HPLC-MS, 1HNMR, Microanalysis.
Solubility: Soluble in DMSO.